Mafuta a Lorcaserin (616202-92-7)

October 30, 2018

Yaikulu ya Lorcaserin ufa ndi wa gulu la mankhwala omwe amadziwika kuti serotonin receptor agonists.Igwira ntchito powonjezera kukhudzika kwakumverera kotero kuti …… ..


Chikhalidwe: Mu Kupanga Misa
Unit: 25kg / Drum
mphamvu: 1480kg / mwezi

Vuto lakuda la Lorcaserin powder (616202-92-7) kanema

 

Mafinya a Lorcaserin powder (616202-92-7) Kufotokozera

Nkhungu ya Lorcaserin ndi ya mankhwala omwe amadziwika kuti serotonin receptor agonists.Imagwira ntchito poonjezera chidziwitso chokwanira kuti chakudya chochepa chidyedwe.Raw Lorcaserin powder amagwiritsidwa ntchito ndi ntchito yovomerezedwa ndi dokotala, kusintha kwa khalidwe, komanso pulogalamu ya zakudya zowonongeka kukuthandizani kuchepa thupi. Amagwiritsidwa ntchito ndi anthu ena olemera kwambiri, monga omwe ali olemera kwambiri kapena odwala matenda okhudzana ndi kulemera. Kutaya thupi ndi kuzisiya kungachepetse mavuto ambiri azaumoyo omwe amabwera ndi kunenepa kwambiri, kuphatikizapo matenda a mtima, shuga, kuthamanga kwa magazi, ndi moyo wautali.

Mafuta a Lorcaserin ndi 5-HT2C receptor agonist, ndipo kuyesa kwa vitro kwa mankhwalawa kunawonetsa kusankha kwa 5-HT2C pazolinga zina zokhudzana nazo. 5-HT2C zolandilira zimapezeka pafupifupi muubongo wokha, ndipo zimapezeka mu choroid plexus, kotekisi, hippocampus, cerebellum, amygdala, thalamus, ndi hypothalamus. Kukhazikitsa kwa 5-HT2C receptors mu hypothalamus ikuyenera kuyambitsa kupanga kwa proopiomelanocortin (POMC) ndipo chifukwa chake kumalimbikitsa kuchepa thupi kudzera kukhuta. Kafukufuku wamankhwala akuwonetsa kuti mankhwalawa amatha kuchepetsa kunenepa kwambiri komanso odwala onenepa kwambiri, amatha kusintha magawo am'magazi okhudzana ndi kunenepa kwambiri, ndipo amalekerera bwino. Mafinya a Lorcaserin oyandikana nawo 5-HT2c nthawi 100 kuposa 5-HT2B (chiwopsezo cha matenda a mtima wa valvular), chimakhala ndi chitetezo chabwino, ndi mankhwala oyamba ovomerezeka ochepetsa thupi pambuyo pa 1999. M'chaka cha Raw Lorcaserin ufa wothira, kuchepa kwakanthawi kochepa kuyambira 3 mpaka 3.7 peresenti.

 

Mpweya wambiri wa Lorcaserin (616202-92-7) Szizindikiro

Name mankhwala Yaikulu Lorcaserin powder Base
Mankhwala Name Raw Lorcaserin powder;(R)-8-Chloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine
Brand NAme Belviq
Kalasi ya Mankhwala serotonin receptor agonists
Nambala ya CAS 616202-92-7
InChIKey XTTZERNUQAFMOF-QMMMGPOBSA-N
Maselo Fmphutsi C11H14ClN
Maselo Wasanu ndi atatu 195.69
Misa ya Monoisotopic 195.0814772
Kusungunula Pmafuta  Palibe deta yomwe ilipo
Fkubwezeretsanso Pmafuta Palibe deta yomwe ilipo
Halimo Half-Life Malasita theka la moyo ndi maola pafupifupi 11.
mtundu White powder
Kutupa  Kutentha kwa madzi kumaposa 400 mg / mL.
yosungirako Tkutentha  -20 ℃ Freezer
Amalingaliro Kuchepetsa kunenepa kwambiri, monga kulongosola zakudya zopereŵera-calorie ndi kuchulukitsa zochitika za thupi.